ACTIVE PHARMACEUTICAL INGREDIENTS


 

INGREDIENT

CAS #

ACTIVITY

5-Flucytosine

2022-85-7

Antimetabolite, Antifungal

8-Chlorotheophylline 85-18-7

mild central nervous system stimulant, Purine

Abacavir

136470-78-5

Anti-HIV agent, Nucleoside and Nucleotide Reverse Transcriptase inhibitor

Abaperidone

183849-43-6

 

Abarelix

183552-38-7

Antineoplastic agent, Anti-Testosterone agent

Abciximab

143653-53-6

Anticoagulant, Antiplatelet agent

Abetimus

167362-48-3

 

Abrineurin

178535-92-7

Treatment of amyotrophic lateral sclerosis

Acamprosate

77337-76-9

Alcohol Deterrent

Acarbose

56180-94-0

Hypoglycemic agent, Alpha-glucosidase inhibitor

Aceclofenac 89796-99-6

 

Acetaminophen

103-90-2

Analgesic

Acetazolamide

59-66-5

Diuretic, Anticonvulsant, Carbonic Anhydrase inhibitor

Acetophenazine

2751-68-0

Antipsychotic

Acetylsalicylic Acid

50-78-2

Fibrinolytic agent, Antiinflammatory agent, Anticoagulant

Aciclovir 59277-89-3 Antiviral
Acipimox51037-30-0

 

Acitretin55079-83-9

 

Acrosoxacin

40034-42-2

Antiinfective, Quinolone antibiotic

Actinomycin

50-76-0

Polypeptide antibiotic, Antibacterial agent, Antineoplastic agent

Adalimumab

331731-18-1

Immunomodulatory agent, Antirheumatic agent

Adamantane 281-23-2

 

Adapalene106685-40-9 Anti-acne agent, similar to Vitamin A;
Adefovir Dipivoxil142340-99-6

 

Adefovir 106941-25-7 nucleotide analogue reverse transcriptase inhibitor (NtRTI),

Adenosine

58-61-7

Vasodilator agent, Antiarrhythmic agent, Analgesic, Cardiac

Adinazolam

37115-32-5

Antidepressant

Adrogolide

171752-56-0

 

Agalsidase Alfa

104138-64-9

Treatment of Fabry Disease.

Agalsidase Beta

104138-64-9

Enzyme replacement

Albendazole 54965-21-8

 

Albuterol

18559-94-9

Tocolytic agent, Bronchodilator agent

Aldesleukin

85898-30-2

Antineoplastic agent

Alefacept

222535-22-0

Treatment of plaque psoriasis

Alefacept

222535-22-0

Immunomodulatory agent, Immunosuppresant

Alemcinal

150785-53-8

 

Alendronate Sodium121268-17-5 bisphosphonate drug to treat osteoporosis

Alendronate

66376-36-1

Antiresorptive, Bisphosphonates

Alfentanil

71195-58-9

Anesthetic, Narcotic, Analgesic, Opiate agonist

Alfuzosin

81403-80-7

Antihypertensive agent

Alglucerase

37228-64-1, 143003-46-7

Enzyme replacement

Alibendol 26750-81-2

 

Alitretinoin

5300-03-8

Antineoplastic used in the treatment of AIDS-related Kaposi's sarcoma and in the treatment of acute promyelocytic leukemia

Alitretinoin

5300-03-8

Antineoplastic agent

Allopurinol

315-30-0

Free Radical Scavenger, Enzyme inhibitor, Antimetabolite, Gout Suppressants

Almitrine Mesylate

27469-53-0

Respiratory agonist

Almotriptan

181183-52-8

Anti-migraine agent, Antiinflammatory agent, Vasoconstrictor agent, Selective Serotonin agonist

Alosetron

122852-42-0

Gastrointestinal agent, Serotonin 5-HT3 receptor antagonist

Alpha-1-proteinase Inhibitor

9041-92-3

Enzyme

Alprazolam

28981-97-7

Antianxiety agent, benzodiazepine anticonvulsant, antianxiety agent, muscle relaxant

Alprazolam-d5 125229-61-0 benzodiazepine anticonvulsant, antianxiety agent, muscle relaxant

Alprenolol

13655-52-2

Sympatholytic, Antihypertensive agent, Antiarrhythmic agent

Alteplase

105857-23-6

Thrombolytic agent

Altinicline

179120-92-4

 

Altretamine

645-05-6

Antineoplastic agent

Aluminium Glycinate 13682-92-3

 

Aluminum Hydroxide 21645-51-2

 

Alvameline

120241-31-8

 

Ambenonium

7648-98-8

Antiarrhythmic agent, Antimyasthenics

Ambroxol Hydrochloride 23828-92-4

 

Amediplase

151912-11-7

 

Amfebutamone 34911-55-2

 

Amifloxacin Mesylate

88036-80-0

Quinolone antibiotic
Amifloxacin

86393-37-5

Quinolone antibiotic

Amifostine

20537-88-6

Radiation-Protective agent

Amiglumide

119363-62-1

 

Amikacin Sulfate 39831-55-5

Antibacterial agent, Aminoglycoside

Amikacin

37517-28-5

Antibacterial agent, Aminoglycoside

Aminoglutethimide

125-84-8

Antineoplastic agent, Adrenergic agent

Aminophylline 317-34-0

 

Aminophylline

317-34-0

Cardiotonic agent, Bronchodilator agent, Respiratory Smooth Muscle relaxant

Aminosalicylic Acid

65-49-6

Antituberculosis agent

Amiodarone Hydrochloride 199774-82-4

 

Amiodarone

1951-25-3

Vasodilator agent, Antiarrhythmic agent, Antiarrhythmic agent

Amitivir

111393-84-1

 

Amitriptyline

50-48-6

Analgesic, Antidepressant, Norepinephrine-Reuptake inhibitor

Amlodipine Maleate88150-47-4

Vasodilator agent, Antianginal, Antihypertensive agent, Calcium Channel Blockers

Amlodipine

88150-42-9

Vasodilator agent, Antianginal, Antihypertensive agent, Calcium Channel Blockers

Amodiaquine Dihydrochloride6398-98-7

 

Amodiaquine86-42-0

 

Amorolfine 78613-35-1

 

Amoxapine

14028-44-5

Antidepressant, Norepinephrine-Reuptake inhibitor

Amoxicillin

26787-78-0

Antibacterial agent

Amoxicillin

26787-78-0

 

Amphetamine

300-62-9

Adrenergic agent, Dopamine agent, Central Nervous System agent

Ampicillin Sodium

69-52-3

 

Ampicillin Trihydrate

7177-48-2

 

Ampicillin

69-53-4

Antibacterial agent

Ampiroxicam99464-64-9

 

Amprenavir

161814-49-9

Antiviral, HIV protease inhibitor

Amprenavir

161814-49-9

Anti-HIV agent, Antibiotic

Amprenavir

161814-49-9

 

Amrinone 60719-84-8

 

Amsacrine

51264-14-3

Antineoplastic agent

Anagrelide Hydrochloride

58579-51-4

 

Analgin68-89-3

 

Anastrozole

120511-73-1

Antineoplastic agent

Ancestim

163545-26-4

Treatment of anemia; hematopoietic adjuvant, stem cell factor

Anecortave Acetate

7753-60-8

Treatment of diseases involving neovascularization of the eye, angiostatic steroid

Anethol Trithion 532-11-6

 

Anidulafungin

166663-25-8

Antifungal used in the treatment of infections caused by Candida, allspecies

Anileridine

144-14-9

Analgesic, Narcotic, Opiate agonist

Aniprime2135-17-3

 

Aniracetam 72432-10-1

 

Anisperimus

170368-04-4

 

Anistreplase

81669-57-0

Thrombolytic agent

Apalcillin

63469-19-2

 

Apomorphine

41372-20-7

Antiparkinson agent, Dopamine agonist

Apraclonidine

66711-21-5

Antiglaucomic agent, Ophthalmic

Aprepitant

170729-80-3

Antiemetic in chemotherapy-induced emesis; antidepressant; treatment of psychiatric conditions

Aprepitant

170729-80-3

Antiemetic

Arbekacin

51025-85-5

 

Arcitumomab

154361-48-5

Diagnostic agent, Imaging agent

Argatroban

74863-84-6